[HN Gopher] HIV in cell culture can be completely eliminated usi...
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       HIV in cell culture can be completely eliminated using CRISPR-Cas
       gene editing [pdf]
        
       Author : geox
       Score  : 290 points
       Date   : 2024-03-19 23:12 UTC (23 hours ago)
        
 (HTM) web link (www.escmid.org)
 (TXT) w3m dump (www.escmid.org)
        
       | eganist wrote:
       | Way out of my depth here, but I'm guessing the main hurdles to
       | turning this into a drug are encapsulation in a way that survives
       | injection (or better yet, ingestion) as well as either targeting
       | of infected cells or at least ensuring that even if it touches
       | every cell, it only affects HIV DNA?
       | 
       | Basically, what's needed to commercialize this?
        
         | colechristensen wrote:
         | crispr also makes mistakes. The kind that lead to cancer,
         | disability and death. It's not a magic wand. Being able to do
         | something in cell culture is interesting but very far away from
         | a therapy.
        
           | smt88 wrote:
           | How do Casgevy and Lyfgenia[1] avoid these dangerous
           | mistakes? Is it something that can be generalized to other
           | therapies, or does it need to be recreated for each "edit"
           | that we want to turn into a therapy?
           | 
           | 1. https://www.fda.gov/news-events/press-announcements/fda-
           | appr...
        
             | ghkbrew wrote:
             | According to your link, both of those are applied to
             | extracted stem cells which are then reintroduced. The
             | ability to perform clonal expansion and DNA sequencing
             | makes it possible that screening for off-target edits could
             | be performed. Though I have no idea if it's actually done.
        
           | jryb wrote:
           | Your point is broadly correct (not sure about disability
           | though), but I think it overstates the danger of what will
           | happen in practice. Yes, if you picked a random target and
           | blasted away, you probably wouldn't have a good time. But
           | anything that even approaches clinical trials is going to get
           | substantial engineering put into it to minimize (and
           | characterize) all of the off-target loci. If there's
           | meaningful editing near an oncogene then that's going to be a
           | deal breaker for a particular guide. When the FDA was
           | discussing the Casgevy application, they went into remarkable
           | detail of how Vertex had measured the off-targets - the
           | regulators really, really don't want to approve anything
           | risky.
           | 
           | Frankly just getting it to work at all is the real hurdle in
           | this case.
        
             | _heimdall wrote:
             | > If there's meaningful editing near an oncogene then
             | that's going to be a deal breaker for a particular guide.
             | 
             | At this point do we know every gene that had the potential
             | to cause cancer?
        
               | a_bonobo wrote:
               | We roughly know the space of possible mutations in the
               | human genomes because we have so many sequenced genomes
               | now: if we don't spot a mutation it's probably not good
               | when it happens, survivorship bias.
               | 
               | The problem with CRISPR is that we cannot control _where_
               | the off-target effects happen, we can currently only
               | optimise the guiding RNA and the Cas enzyme to have as
               | little off-target effects as possible (but not 0, yet).
               | It would be cool to engineer guiding RNAs that bind in
               | those high mutation-rate areas when they have off-target
               | effects, stuff can mutate there and nothing will happen
               | (probably).
        
             | colechristensen wrote:
             | > Frankly just getting it to work at all is the real hurdle
             | in this case
             | 
             | This being the point. Many diseases have been cured dozens
             | of times over in a tissue sample in a lab that never make
             | it to actual therapies because the hurdle is elsewhere. The
             | risks with crispr are as stated, especially flooding your
             | entire body with it to target a virus.
        
             | AllegedAlec wrote:
             | > Your point is broadly correct (not sure about disability
             | though), but I think it overstates the danger of what will
             | happen in practice
             | 
             | https://www.nature.com/articles/nrc1122
        
             | amluto wrote:
             | One thing I was confused by: why did Vertex choose to
             | reactivate HbF instead of attempting to correct the
             | mutation that causes sickle cell disease in the first
             | place?
        
               | bglazer wrote:
               | CRISPR, in the form used by Vertex, is not capable of
               | directly repairing an existing gene. In the case of
               | sickle cell this means directly changing the mutated
               | nucleotide in the HbA gene. CRISPR is very capable of
               | _cutting_ the genome at precise locations. These cuts
               | lead to lossy repair pathways that introduce mutations or
               | deletions that disable the gene at the spot that CRISPR
               | cut. So, the best you can hope for is that the CRISPR cut
               | leads to a loss of function. It 's possible to use CRISPR
               | to introduce new sequences into the DNA, by introducing a
               | new DNA sequence alongside the CRISPR proteins, then
               | hoping that DNA repair "accidentally" uses the genetic
               | sequence you put in to repair the break in the DNA. This
               | is even less efficient than just cutting the DNA, and it
               | would not fix the mutated HbA, so it's not really
               | therapeutically relevant for sickle cell.
               | 
               | There are more recent techniques, notably prime editing,
               | that use a modified version of the CRISPR system that can
               | introduce changes to single bases (nucleotides) in the
               | genome. These have some promise of directly fixing
               | diseases caused by single mutations, but there are
               | hurdles in terms of efficiently delivering the prime
               | editor to the right tissues as well as efficiency of the
               | actual repair.
        
               | amluto wrote:
               | So how is Vertex activating HbF? Did they find some bases
               | to remove that cause the gene to be expressed more than
               | usual?
        
         | aaauaucuggaa wrote:
         | Generally speaking:
         | 
         | - Delivery: getting the mRNA and guide RNA into the target
         | cells
         | 
         | - Expression: ensuring the target cell expresses the mRNA, thus
         | making the protein
         | 
         | - On Target Editing Efficiency: ensuring the intended edit
         | happens at a high rate
         | 
         | - Off Target Editing: ensuring other edits in other locations
         | do not occur
        
         | nextaccountic wrote:
         | Does this means that in order to productionize this into a
         | drug, one would need to basically engineer a biological virus?
        
           | jjtheblunt wrote:
           | https://en.wikipedia.org/wiki/Viral_vector
        
             | lucioperca wrote:
             | or mRNA
        
               | XorNot wrote:
               | CRISPR is pretty complicated - I'd say it's not clear
               | whether mRNA of such length could stably produce enough
               | enzyme in enough places. It's great when you need an
               | antigen to be presented, but not so much when you need an
               | entire restriction enzyme system.
        
         | WheelsAtLarge wrote:
         | There's a sickle cell therapy that uses CRISPR. I don't know
         | the specifics but if one has been successful then a second can
         | be too. I'm looking forward to getting more information in the
         | future. Cell culture vs cure is a long road but at least
         | there's hope. The big drawback is that these therapies are
         | super expensive but time and experience in the past have proven
         | that the costs can be lowered.
         | 
         | "Sickle Cell Disease Approvals Include First CRISPR Gene
         | Editing Therapy"
         | 
         | https://jamanetwork.com/journals/jama/article-
         | abstract/28137....
        
           | crakenzak wrote:
           | Yup Casgevy & Lyfgenia! These sickle cell (and now also
           | approved for beta thalassemia) CRISPR therapies basically
           | work in the following way:
           | 
           | - Blood stem cells are removed from the patient and the
           | CRISPR Cas9 protein outside of the body is injected to cut
           | the gene responsible for suppressing fetal hemoglobin
           | production (even people with sickle cell have healthy fetal
           | hemoglobin, their adult hemoglobin gene is what causes the
           | deformed red blood cells)
           | 
           | - Chemotherapy is used to kill all living bone marrow and
           | remove all previous unedited stem cells.
           | 
           | - New edited stem cells are inserted, and patient recovers
           | with new blood production being of healthy red blood cells.
           | 
           | I'd say a huge step forward was FDA and EMA approval, but
           | figuring out a way to remove previous unedited stem cells
           | with chemotherapy would be a step change in the patient
           | experience.
        
             | Etheryte wrote:
             | It's both extremely sci-fi and incredibly terrifying that
             | one of the steps for a cure is to quote unquote kill all
             | living bone marrow. Modern medicine is fascinating in how
             | advanced it can be.
        
               | l33tman wrote:
               | Yeah it's a spectacular transplant procedure, though it's
               | really not that modern medicine, it has been developed
               | since the 50s! The step where you irradiate or apply
               | chemo to kill off the existing bone marrow had to be done
               | at first because the patients had leukemia so you had to
               | do this anyway. An interesting thing is that if there are
               | still cells left in you, they will be wiped clean by the
               | new transplanted immune system in a so called graft-vs-
               | host response that also sounds like a horror-movie
               | concept :)
        
               | renegade-otter wrote:
               | And yet, measles are back.
        
               | blkhawk wrote:
               | not sure if you need to kill absolutely all living bone
               | marrow. Unlike cancer having 5% sickle cell red blood
               | cells is probably fine. That makes the chemo probably way
               | less bad than what you would need for cancer.
        
             | giantg2 wrote:
             | "- Chemotherapy is used to kill all living bone marrow and
             | remove all previous unedited stem cells.
             | 
             | - New edited stem cells are inserted, and patient recovers
             | with new blood production being of healthy red blood
             | cells."
             | 
             | It's very likely HIV could be cured similarly. I believe
             | all the people who have been cured so far are bone marrow
             | transplant recipients in which the marrow had a specific
             | gene or genes.
        
           | saati wrote:
           | It's very different, you only have to fix some of the bone
           | marrow to help someone with sickle-cell, but you have to
           | eliminate all reservoirs of HIV to cure AIDS.
        
             | WheelsAtLarge wrote:
             | I was under the understanding that HIV attacks only immune
             | cells, white blood cell, only. All the issues that
             | eventually kill are due to the body not being able to
             | defend itself. So it seems like a cure would be very much
             | similar to a sickle cell cure. Is that not the case?
        
           | dghughes wrote:
           | A good video explanation of that too via Sci Show. It's quite
           | complex; chemo, lab work and takes a long time and not always
           | successful but the majority of the time it is successful.
           | 
           | https://www.youtube.com/watch?v=uHWD8RSw4As
        
       | notfish wrote:
       | Relevant xkcd http://xkcd.com/1217
        
         | stared wrote:
         | Actually, a handgun is unlikely to kill bacteria.
        
           | croemer wrote:
           | It's a joke, also the xkcd talks about cancer cells, not
           | bacteria
        
       | ngcc_hk wrote:
       | Is it the greatest day or the worst day (or both at the same
       | time) of humanity when CRISPR is invented ?
        
         | wigster wrote:
         | probably great for humanity 2.0
         | 
         | amazing and scary stuff
        
         | passwordoops wrote:
         | Like nuclear
        
         | epgui wrote:
         | Probably not "the greatest day", but definitely a very very
         | good day.
         | 
         | I think it's too easy to imagine Orwellian scenarios, but I
         | think the real worries are much more subtle than people usually
         | think, and they usually have more to do with how the world
         | already works than with how it could change.
        
         | kjkjadksj wrote:
         | We had the ability to do what crispr did already, it just
         | simplified the lab work. See TALEN and zinc finger nucleases.
        
       | Khelavaster wrote:
       | You'd hope so.. the treatment is already in phase 1/2 combined
       | human trials!
       | 
       | https://crisprmedicinenews.com/news/clinical-trial-update-po...
        
       | Metacelsus wrote:
       | The big problem is that the CRISPR would need to be delivered to
       | 100% of infected cells. And as far as I know (I'm a biologist)
       | nobody has a method that can achieve a delivery rate of 100% in
       | vivo.
        
         | cft wrote:
         | That would be for a cure, but not for a recurrent therapy
        
           | mlrtime wrote:
           | Do we even need a cure or therapy if we can essentially use
           | this as a vaccine?
           | 
           | Doesn't help people now, but may eliminate it as a threat for
           | future generations.
        
             | huytersd wrote:
             | Well you can't use it as a vaccine since there would be no
             | hiv to preemptively excise.
        
           | ac2u wrote:
           | Could that risk evolutionary pressure on whatever is left
           | behind so that mutations emerge that are more aggressive?
        
             | SketchySeaBeast wrote:
             | If we assume that the treatment needs to reach the HIV cell
             | to effect it, and that the danger is not 100% of the cells
             | are reached, would it produce evolutionary pressure? The
             | survivors aren't interacting with whatever got its buddies,
             | right?
        
               | simcop2387 wrote:
               | That itself is an evokutionary pressure. Whatever allowed
               | them to get missed would get amplified by reproduction.
               | Only if it's entirely utterly and only random chance and
               | not something like the method doesn't target certain
               | cells would it not be applying pressure
        
               | yau8edq12i wrote:
               | If you bomb a cow pasture with napalm, you aren't going
               | to be left with napalm resistant cows. Just lucky ones.
               | And luck isn't genetic.
        
               | ac2u wrote:
               | You're viewing the cows in isolation here. Replace the
               | cows with cancer cells with different mutations and it
               | doesn't work anymore.
               | 
               | There's research going with certain types of cancer where
               | the doses of cancer-killing drugs isn't intended to
               | eradicate all cancer cells, but to keep it at a level
               | that's manageable with future treatments.
               | 
               | The theory being that if you go too far, cells that are
               | left with a "lucky" mutation can grow without
               | competition, leaving the patient in an even-less
               | treatable state down the line.
        
               | yau8edq12i wrote:
               | ... Cancer cells? This is about HIV. What are you talking
               | about?
        
               | ac2u wrote:
               | you're talking about cows in a HIV discussion, so I could
               | have said "cows and napalm? we're talking about HIV!",
               | but I'm charitably engaging with your analogy to show
               | that evolutionary pressure is an active research area in
               | disease treatment.
        
             | throwawaymaths wrote:
             | The selection pressure would have to be some form of
             | resisting the crispr tools from entering the cell or
             | functioning in the cell.
             | 
             | The HIV genome is small and I would be surprised if it were
             | so easy for such a thing to come about.
        
               | ac2u wrote:
               | I'm thinking more of a mutation already present that has
               | less treatable traits but can't spread because
               | neighbouring cells are already infected. But then when
               | the treatment is delivered, it isn't cleared because of
               | the difficulty of the delivery mechanism, but the
               | treatment _does_ clear up the surrounding cells,
               | providing fresh ground for the mutated strain to
               | reinfect.
               | 
               | (This is an active research area I've read about in
               | cancer treatment, where it's been suggested that being
               | too aggressive with clearing certain cancers encourages
               | reservoirs of already mutated aggressive variants to be
               | unleashed after treatment whereas before the avenues they
               | had to spread were already infected with the less
               | aggressive variant).
        
               | tg180 wrote:
               | ... and so?
               | 
               | Evolutionary pressure is present in any situation and is
               | unavoidable. It still has an effect even in cases where
               | treatments are effective with a success rate of 100%: the
               | selection of diseases for which there is no cure.
               | 
               | Entertaining such a perspective can lead to an extreme
               | and undesirable conclusion, that the only logical outcome
               | is to do nothing and dismantle the entire modern medical
               | practice.
               | 
               | It's not very constructive.
        
         | m3kw9 wrote:
         | Does it need to be 100%? We have dormant viruses that are
         | domant and would only activate when conditions are good, like
         | colds, and we have ways to deal with it. It's an analogy, for
         | aids we would deal with it with meds and press it back there by
         | turning it into a sort of nuisance like colds. The issue is
         | cost and stigma of passing it. I for one still wouldn't want
         | aids to be as prevalent as the cold even if it's super easy to
         | deal with.
        
         | huytersd wrote:
         | There are specific latent reservoirs the HIV hides in. It
         | wouldn't need to get every cell in the body, just have a
         | favorable probability distribution to hit the reservoirs.
        
       | croemer wrote:
       | Science by press release. The results aren't even preprinted yet.
       | Only some methods in a 2022 preprint. Looks hyped up, I'd ignore.
       | 
       | > This press release is based on abstracts P0004 P0006, P0013,
       | P0026 and P0004 at the European Congress of Clinical Microbiology
       | & Infectious Diseases (ECCMID). The material has been peer
       | reviewed by the congress selection committee. Only material from
       | P0004 has been published in a preprint article. The other three
       | have not yet been submitted to a medical journal or as preprints.
        
       | slackfan wrote:
       | You can also eliminate most climate-change-causing pollution (and
       | microplastics) via nuclear weapons.
        
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