[HN Gopher] Phenethylamines I have feared and loathed (2020)
       ___________________________________________________________________
        
       Phenethylamines I have feared and loathed (2020)
        
       Author : kvee
       Score  : 70 points
       Date   : 2022-02-06 09:18 UTC (2 days ago)
        
 (HTM) web link (nikobidin.com)
 (TXT) w3m dump (nikobidin.com)
        
       | perardi wrote:
       | Not mentioned in the post, but mentioned in the book that
       | inspired the post:
       | 
       | 2C-B is a fun one. Good times have been had there.
        
         | c7DJTLrn wrote:
         | Seemed overrated to me. Maybe I got the dose wrong but the
         | purity can be so inconsistent that everyone's going to have a
         | different experience. I'd much rather take some classic LSD,
         | you know what you're in for and it doesn't end disappointingly
         | early like 2C-B.
        
           | capableweb wrote:
           | 2C-B has a very "surface level" high compared to LSD, which
           | can absolutely make your mind go into itself, 2C-B doesn't
           | take itself as serious. 2C-B can be fun even in larger groups
           | where you don't know people too well, and it's mostly just
           | visual gags and euphoria that happen. LSD on the other hand
           | requires a personal connection to everyone in the group
           | already, triggers deep introspection and is not nearly as
           | visual as 2C-B, and euphoria only happens when it would
           | happen in real-life, but LSD can easily make you go down the
           | other road.
        
           | netizen-936824 wrote:
           | 2C-B was enjoyable but seriously lacks introspection from my
           | experience. It felt like "psychedelic-lite" where the visual
           | effects are quite pronounced... but that's about it
           | 
           | LSD is a different ballgame from the 2C family IMO, its
           | difficult to compare. From my experience (again this is quite
           | subjective) the visuals from LSD weren't as "thick" and
           | deeply colorful. They had a sort of whispyness to them and
           | (usually) a much deeper headspace
        
             | oceanghost wrote:
             | > the visual effects are quite pronounced
             | 
             | This is what I remember about 2CB. It looked like the
             | Matrix effect to me but in translucent rainbow colors.
        
           | loves_mangoes wrote:
           | I'm surprised, because you don't often hear that particular
           | criticism of 2C-B. Mostly, people complain about nausea, or
           | the fact that it burns very painfully when people insuflate
           | it
           | 
           | Purity and accurate dosage is a function of your vendor.
           | Buying 2C-B pills will be more dangerous, they are
           | notoriously underdosed and should ideally be sent to a lab
           | first, but at the very least spot-checked with a reagent test
           | kit.
           | 
           | Duration is a subjective preference, I feel. LSD is nice, I
           | like it very much, but I can understand than 12 hours
           | uninterrupted is not something everyone can allocate in their
           | schedule.
        
             | c7DJTLrn wrote:
             | Yep, I spared the details regarding nausea but the contents
             | of my stomach were definitely emptied once or twice. As far
             | as I remember it wasn't anything special and the additional
             | side effects and risk you describe make it just not worth
             | it in my opinion.
        
               | Scoundreller wrote:
               | > I spared the details regarding nausea but the contents
               | of my stomach were definitely emptied once or twice.
               | 
               | Zofran works for my friend, zofran. Whether it's specific
               | serotonin blocking effects that fixes the nausea has +/-
               | psych experience is unknown.
               | 
               | (Supposedly it can contribute to serotonin syndrome, but
               | I don't understand the mechanism. Seems theoretical, but
               | don't say I didn't warn you).
        
               | loves_mangoes wrote:
               | That's fair enough. I did hear it repeated a lot that
               | 2C-B's dosage curve seems to be particularly steep and
               | non-linear. I don't know that it's been studied very
               | scientifically, but reportedly the difference between 40
               | and 50mg is much bigger than the difference between 20
               | and 30.
               | 
               | I stick to low dosages, partly to avoid nausea and partly
               | because I like to be somewhat cautious with this delicate
               | biological machinery I don't understand.
               | 
               | For me it's also something I can take a small dose of
               | occasionally when I have a big night out, if I'd like to
               | sleep early, or if I'd like more stimulation and less
               | headspace.
               | 
               | LSD I use for long introspective trips, physically by
               | myself so that I can tune in and out of online social
               | interactions depending on how I feel.
               | 
               | I feel like 2C-B is a nice option to have for different
               | settings. Since I don't very much experience the
               | downsides it's worth it for me, but I can definitely
               | acknowledge the downsides =)
        
         | pmoriarty wrote:
         | _" Not mentioned in the post, but mentioned in the book that
         | inspired the post: 2C-B"_
         | 
         | It is mentioned in the article:
         | 
         |  _" these and other reasons make me suspect that even 'safer'
         | phenethylamines like 2C-B won't be getting FDA approval anytime
         | soon."_
        
         | dr_dshiv wrote:
         | One can write fluently on half a pill, which is quite handy.
        
       | capableweb wrote:
       | The author mentions that 2C-P has "notable physical discomfort"
       | and I can attest to that, although I didn't have effects for as
       | long as stated (my trip was more around 7-8 hours, author states
       | "up to 20 hours", and my onset was also faster) it had a
       | significant discomfort, especially when compared to 2C-B which
       | induces a loud, unstoppable euphoria. It wasn't as much of a
       | physical discomfort but a mental one. Eventually what calmed me
       | down from the 2C-P was watching a newly released movie I never
       | really bothered paying attention to before, Avatar.
       | 
       | None the less, interesting to see this list on HN, and read about
       | some new compounds I haven't heard about before (hello
       | 25B-NBOMe).
        
         | tepitoperrito wrote:
         | I'd stay far away from any compound in the 25x-NBOMe series.
         | The risk of life threatening episodes are real and understated
         | in TFA with erratic responses to even low doses in experienced
         | and first time users.
         | 
         | One summer when 25i first hit the scene SWIM was taking 1000 to
         | 5000 microgram doses weekly until one week SWIM dosed 1000
         | micrograms (pre dipped blotter) and the short version of the
         | story is SWIM woke up in the hospital and was being monitored
         | to prevent kidney failure due to elevated proteins in SWIM's
         | blood.
         | 
         | Similar events which were all preceded by psychotic breaks with
         | reality happened to quite a few of SWIM's friend group if you
         | want some anecdata to add there.
         | 
         | It's scary stuff whose unpredictability means I wouldn't
         | recommend touching it with a 10 foot pole.
        
       | philipkglass wrote:
       | This post was a real trip down memory lane, back to the days of
       | The Hive [1].
       | 
       | Before Shulgin published _Phenethylamines I Have Known and Loved_
       | and _Tryptamines I have Known and Loved_ , Donald Cooper of the
       | Drug Enforcement Administration wrote this prescient 1988
       | document titled "Future Synthetic Drugs of Abuse":
       | 
       | https://erowid.org/library/books_online/future_synthetic/fut...
       | 
       | It's like looking into the 2000s from a vantage point of the
       | 1980s. What was really necessary for wild and woolly synthetic
       | drugs to take off was digital infrastructure. That is, tools for
       | collaborative and secret discussion, research tools [2], and
       | (more recently) darknets.
       | 
       | The thing that finally made me stop following the scene was that
       | I liked the _how-to_ hacking aspect of the chemistry. There were
       | tons of threads about how to make equipment, source chemicals
       | from unexpected places, and synthesize the critical intermediates
       | that were on watch-lists so they were difficult /inadvisable to
       | buy commercially.
       | 
       | The last forum I followed closely ("Blacklight") ended up with
       | members just theorizing about interesting points in chemical
       | space and then outsourcing the manufacturing to commercial
       | contract labs, mostly in China [3]. The only actual chemistry
       | that would be done outside China was instrumental analysis (to
       | confirm composition/purity of products). And the scene became
       | secretive and scheming about people spotting chemicals that were
       | subjectively good enough to become popular and commercializing
       | them in Europe before the law caught up. (It's globalization in
       | miniature! Keep marketing and management domestic, but offshore
       | the low margin manufacturing work.)
       | 
       | The Hive wasn't like that. Most of the chemicals the members
       | wanted to make were old stalwarts -- amphetamine,
       | methamphetamine, MDA, and MDMA were the most popular. All the
       | close analogs were illegal already so members were united in
       | finding ways to hack around the restrictions. Nobody expected to
       | hack around the law itself, i.e. to escape without consequences
       | if the law caught them with the output of their clandestine labs.
       | All questions that indicated someone was trying to scale up to
       | major commercial manufacturing would get banned anyway. So users
       | were generally collaborative rather than competitive. Everyone
       | would pitch in on e.g. trying to figure out how to remove pill
       | binders from OTC decongestants so that the purified
       | pseudoephedrine was suited for downstream transformation to
       | methamphetamine. Even people who wanted to manufacture less
       | popular or more obscure compounds really wanted to do it in their
       | own garage -- not in a contract lab.
       | 
       | [1] https://web.archive.org/web/20040103031950/http://the-
       | hive.w...
       | 
       | [2] Back when The Hive was active, there were huge ongoing
       | request threads for people trying to source research papers.
       | Other members would have to go to a library, photocopy articles
       | from the stacks, and upload scans. It was a huge breakthrough
       | when the American Chemical Society actually scanned its complete
       | print run and made those available to subscribers online; then
       | members could just download requested papers from their
       | company's/university's account. Then sci-hub solved even the part
       | where someone has to manually request a paper.
       | 
       | [3] This preceded the rise of imported fentanyl by several years.
       | In fact I wouldn't be surprised if small time (but technically
       | advanced) Western drug dealers actually kickstarted the trend of
       | getting potent opioids manufactured in China.
        
         | louky wrote:
         | I still miss the hive regularly. So many great discussions lost
         | in the fog.
        
           | philipkglass wrote:
           | In 2015 one of the original admins provided a backup so that
           | a reasonably complete mirror could be hosted on Erowid:
           | 
           | https://www.sciencemadness.org/whisper/viewthread.php?tid=63.
           | ..
           | 
           | https://the-hive.archive.erowid.org/forum/forums.pl
           | 
           | So you can read it again even though none of us can go back
           | in time again.
        
         | rootsudo wrote:
         | Other points of reference would also be rhodium. But you're
         | spot on, it was a magical point of the Internet.
        
           | philipkglass wrote:
           | Rhodium was the university's library. The Hive was the
           | university's classrooms. Or something like that. I think I
           | came across Hyperreal [1] first, by way of my interest in
           | electronic music, which linked to Erowid [2], which led me to
           | Rhodium and the Hive.
           | 
           | As someone fascinated by chemistry since childhood, I was in
           | digital heaven. I was far too risk averse to consider making
           | controlled substances myself, but I loved participating in
           | the publication-sourcing and equipment discussion.
           | 
           | [1] http://hyperreal.org/
           | 
           | [2] https://www.erowid.org/psychoactives/psychoactives.shtml
        
       | netizen-936824 wrote:
       | I would likely agree with all the conclusions here besides one of
       | them. 2C-P is a fascinating compound and while it may be
       | difficult to administer orally in therapy, there may be other
       | viable routes. The subjective headspace of extreme introspection
       | induced by this compound is absolutely incredible and will make
       | you seriously examine how you feel about your self.
        
       | inglor_cz wrote:
       | For anyone who is confused by the title: this is a variation of
       | the book name "Phenethylamines I Have Known and Loved", published
       | by a scientist couple in 1991.
       | 
       | https://en.wikipedia.org/wiki/PiHKAL
        
         | c7DJTLrn wrote:
         | I wish there was something like PIHKAL for non-chemists. I had
         | a fascination for chemistry as a young lad but Shulgin's books
         | are impenetrable for me.
        
           | netizen-936824 wrote:
           | You can just read the subjective reports, those are
           | interesting in their own right.
        
             | pmoriarty wrote:
             | The first part of PiHKAL, written by Ann Shulgin, is also
             | completely non-technical and is a spellbinding story.
             | Highly recommended for anyone interested in the subject
             | matter of the book, whether they know chemistry or not.
        
           | el_benhameen wrote:
           | If you're aware of PIHKAL then you're probably already aware
           | of Erowid, but if not, it's a good source for interesting
           | subjective reports.
        
         | ArnoVW wrote:
         | And "fear and loathing in Las Vegas" I imagine.
         | 
         | https://en.m.wikipedia.org/wiki/Fear_and_Loathing_in_Las_Veg...
        
           | capableweb wrote:
           | Probably referring to the book/novel rather than the movie,
           | as the book is autobiographical in nature and a fascinating
           | read, while the movie is more pure entertainment.
           | 
           | Edit: actually scratch that, I have no idea (obviously) what
           | the author had in mind, and could be either.
        
             | ncmncm wrote:
             | The book had two of the most enduring images in all of
             | modern literature.
             | 
             | The first, that occurs in a Cadillac convertible bombing
             | toward Las Vegas at 90 mph, has the author seeing big
             | black, bat-like things swooping around the car, and
             | choosing not to mention them to his companion: "He'd see
             | them soon enough, poor bastard."
             | 
             | The second is in the lounge of a hotel on the Strip, when
             | the author suddenly realizes that everyone else in the room
             | is a vicious, bloodthirsty reptile, and the whole floor is
             | a puddle of shed blood.
        
             | Zababa wrote:
             | I wouldn't call the movie pure entertainement, quite the
             | opposite. It can be seen as that, but there are a few
             | scenes that really stays with you if you've ever fooled
             | around with drugs. The most obvious ones are when the
             | narrator talks about San Francisco in the 60's, and when he
             | talks about the "fallacy of acid culture" near the end.
             | There's also something to be said about the "white rabbit"
             | scene, though it's hard to put into words.
        
         | [deleted]
        
       | ipnon wrote:
       | The Controlled Substances Act needs a carve out for substances so
       | strange, obscure and nerdy they would never achieve mainstream
       | popularity or public health effects, but that would require drug
       | policy having some character of consistency and reasonability. A
       | cruel joke where you can only laugh to keep from crying!
        
         | netizen-936824 wrote:
         | The Controlled Substances Act really just needs to be entirely
         | rewritten or thrown out altogether. Same with the DEA.
        
       | Jerrrry wrote:
       | 25b was a very commonly found compound in 2012-2014 gen 1 Silk
       | Road era.
       | 
       | A visual, not too uncomfortable cousin of LSD. Except the risk
       | profile was completely different.
       | 
       | 25i, 25c, 25b, 25d nBome's. The "fake acid" that your high school
       | administration actually had a reason to fret about.
       | 
       | Ironically, xanax is what actually should had had the attention.
       | Maybe the high school administration were taking/selling too much
       | Xanax to see the issue.
        
         | dr_dshiv wrote:
         | Xanax is terrifying. Psychedelics I can handle.
        
       | FollowingTheDao wrote:
       | I cannot even eat food high in trace amines or I get anxious as
       | all get out and I am up all night. Seriously, chocolate gives me
       | insomnia. So I have no idea how someone could handle these drugs.
       | 
       | I think this happens to me for two reasons. I am low in BH4 which
       | limits my ability to metabolize amino acids down the common
       | pathway and thinks like phenylalanine get metabolized dow the
       | alternative pathways creating PEA and Tyramine. But also I have
       | the mental illness associated changes in TAAR1 and VMAT1 and
       | VMAT2. (I have schizoaffective Bipolar Disorder.)
       | 
       | I never understood why people would want to take drugs to see the
       | shit and live the suffering I have all my life but that's where
       | we are...
        
         | ipnon wrote:
         | New York is fine for a visit but I'd never want to live there.
        
       | version_five wrote:
       | This is not subject I know anything about, but I just realized
       | that "betaphenethylamine" is (I think) the drug Case is taking in
       | _Neuromancer_ because normal drugs can 't get him high due to a
       | modification in his pancreas. Maybe not entirely accurate vs this
       | list, but William Gibson continues to amaze me with little
       | details like that.
        
       | newbie789 wrote:
       | I'm glad to hear people discussing this! I love how most of the
       | hippies that love "natural psychedelics" have a loophole for LSD.
       | Just because a drug has a precursor found in nature doesn't make
       | the drug itself natural.
       | 
       | As somebody that experimented heavily with psychedelics when I
       | was much younger, my opinion is that the 2C-B/E/I group have
       | definite possible therapeutic value, and the main thing causing
       | stagnation is the ridiculous hippy mindset that it's ~
       | _synthetic_ ~ and therefore bad. It's ridiculous.
       | 
       | Over the past few years it's been interesting watching polite
       | society "discovering" psychedelics. I really can't wait for these
       | people to find the therapeutic value of smoked/IV DMT, especially
       | considering that it's WAY safer than ayahuasca.
       | 
       | I would love to see a study on the possible therapeutic value of
       | dextromethorphan, but as far as I've seen it's not really on the
       | radar. I know it seems weird, but from subjective experience I
       | found it to be very helpful a few times as a teenager. I used to
       | jokingly call it "therapy in a bottle." It's a real shame that
       | most DXM-containing products nowadays in the US come mixed with
       | other compounds that make it dangerous to take at a
       | recreational/therapeutic dose.
        
       | mwattsun wrote:
       | I can't imagine trying unknown drugs on myself. That's so risky.
       | But people did it and found out the hard way like with Bromo-
       | DragonFLY:
       | 
       |  _subjective effects have been described as "like being dragged
       | to hell and back again. Many times. It is the most evil [thing]
       | I've ever tried. It lasted an eternity." Oh and it lasts up to 3
       | days. No gracias._
        
         | loves_mangoes wrote:
         | The way to test these things is by starting with an alergy
         | test, a dose low enough that it definitely won't have any
         | effect, and also definitely will not kill you.
         | 
         | If you feel fine, you wait several days and try a bigger dose,
         | then see if you feel any effects. Stop when it becomes
         | unpleasant or unwise.
         | 
         | This is not safe. There is no safe way to ingest dozens of
         | unknown chemicals. Somehow, chemists like Shulgin show that
         | it's possible to test all those compounds on yourself and still
         | live a long healthy life. Still, I would not recommend tempting
         | fate.
        
         | gpcr1949 wrote:
         | The fatalities with bromo-dragonfly where due to a mix-up on
         | the distribution end, not only because of the inherent danger
         | of the drugs. In fact, the local distributor (known as Haupt
         | RC) in the bromo-dragonfly 2c-b-fly mix-up incident, died
         | himself. Of course, self-titrating new chemicals is not without
         | risk, but Shulgin style careful titrating usually prevents
         | incidents comparable to the bromo-dragonfly one and various
         | other ones (such as unreliable dosing of NBOMe derivatives
         | etc).
        
       ___________________________________________________________________
       (page generated 2022-02-08 23:00 UTC)